Thierry Masquelin : rechercher sur Z-Library

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1

Context Aware Data-Driven Retrosynthetic Analysis

Nicolaou, Christos A., Watson, Ian A., LeMasters, Mark, Masquelin, Thierry, Wang, Jibo

Journal:

Journal of Chemical Information and Modeling

Année:

2020

Fichier:

PDF, 813 KB

2020

2

ChemInform Abstract: Solution- and Solid-Phase Synthesis of Combinatorial Libraries of Trisubstituted 1,3,5-Triazines.

Thierry Masquelin, Nathalie Meunier, Fernand Gerber, Gerard Rosse

Journal:

Année:

1999

Fichier:

PDF, 28 KB

1999

3

ChemInform Abstract: A New General Three-Component Solution-Phase Synthesis of 2-Amino-1,3-thiazole and 2,4-Diamino-1,3-thiazole Combinatorial Libraries.

Thierry Masquelin, Daniel Obrecht

Journal:

Année:

2001

Fichier:

PDF, 33 KB

2001

4

Novel Solution- and Solid-Phase Syntheses of Heterocyclic Systems

Gaelle Cabon, Berangere Gaucher, Aline Gegout, Sophie Heulle, Thierry Masquelin

Journal:

Année:

2004

Fichier:

PDF, 54 KB

2004

5

Synthesis of Enantiomerically Pure D- and L-(Heteroaryl)alanines by asymmetric hydrogenation of (Z)-α-amino-αβ-didehydro esters

Thierry Masquelin, Emil Broger, Klaus Müller, Rudolf Schmid, Daniel Obrecht

Journal:

Helvetica Chimica Acta

Année:

1994

Langue:

english

Fichier:

PDF, 1.14 MB

english, 1994

6

Naphthopyranquinone Antibiotics: Novel enantioselective syntheses of frenolicin B and some of its stereoisomers

Thierry Masquelin, Urs Hengartnerb, Jacques Streith

Journal:

Helvetica Chimica Acta

Année:

1997

Langue:

english

Fichier:

PDF, 991 KB

english, 1997

7

A Novel Approach towards 2,3,5-Trisubstituted Thiophenes via tandem Michael addition/intramolecular Knoevenagel condensation

Daniel Obrecht, Fernand Gerber, Daniel Sprengeir, Thierry Masquelin

Journal:

Helvetica Chimica Acta

Année:

1997

Langue:

english

Fichier:

PDF, 410 KB

english, 1997

8

A Novel Solution- and Solid-Phase Approach to 2,4,5-tri- and 2,4,5,6-tetrasubstituted pyrimidines and their conversion into condensed heterocycles

Thierry Masquelin, Daniel Sprenger, Roman Baer, Fernand Gerber, Yves Mercadal

Journal:

Helvetica Chimica Acta

Année:

1998

Langue:

english

Fichier:

PDF, 871 KB

english, 1998

9

Investigation of retention behavior of drug molecules in supercritical fluid chromatography using linear solvation energy relationships

Hai Bui, Thierry Masquelin, Tom Perun, Tom Castle, Jeff Dage, Ming-Shang Kuo

Journal:

Journal of Chromatography A

Année:

2008

Langue:

english

Fichier:

PDF, 570 KB

english, 2008

10

New multi-component reaction accessing 3-aminoimidazo[1,2-a]pyridines

John Schwerkoske, Thierry Masquelin, Tom Perun, Christopher Hulme

Journal:

Tetrahedron Letters

Année:

2005

Langue:

english

Fichier:

PDF, 95 KB

english, 2005

11

Sequential Ugi/Strecker reactions via microwave assisted organic synthesis: novel 3-center-4-component and 3-center-5-component multi-component reactions

Thierry Masquelin, Hai Bui, Bob Brickley, Gregory Stephenson, John Schwerkoske, Christopher Hulme

Journal:

Tetrahedron Letters

Année:

2006

Langue:

english

Fichier:

PDF, 139 KB

english, 2006

12

A new general three component solution-phase synthesis of 2-amino-1,3-thiazole and 2,4-diamino-1,3-thiazole combinatorial libraries

Thierry Masquelin, Daniel Obrecht

Journal:

Année:

2001

Langue:

english

Fichier:

PDF, 86 KB

english, 2001

13

A Novel Solid-Phase Approach to 2,4-Diaminothiazoles

Baer, Roman, Masquelin, Thierry

Journal:

Journal of Combinatorial Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 45 KB

english, 2001

14

A remote-controlled adaptive medchem lab: an innovative approach to enable drug discovery in the 21st Century

Godfrey, Alexander G., Masquelin, Thierry, Hemmerle, Horst

Journal:

Drug Discovery Today

Année:

2013

Langue:

english

Fichier:

PDF, 3.12 MB

english, 2013

15

Lipoamide Channel-Binding Sulfonamides Selectively Inhibit Mycobacterial Lipoamide Dehydrogenase

Bryk, Ruslana, Arango, Nancy, Maksymiuk, Christina, Balakrishnan, Anand, Wu, Ying-Ta, Wong, Chi-Huey, Masquelin, Thierry, Hipskind, Philip, Lima, Christopher D., Nathan, Carl

Journal:

Année:

2013

Langue:

english

Fichier:

PDF, 2.30 MB

english, 2013

16

ESR and X-ray Structure Investigations on the Binding and Mechanism of Inhibition of the Native State of Myeloperoxidase with Low Molecular Weight Fragments

Chavali, Balagopalakrishna, Masquelin, Thierry, Nilges, Mark J., Timm, David E., Stout, Stephanie L., Matter, William F., Jin, Najia, Jadhav, Prabhakar K., Deng, Gary G.

Journal:

Applied Magnetic Resonance

Année:

2015

Langue:

english

Fichier:

PDF, 1.57 MB

english, 2015

17

Discovery of selective RIO2 kinase small molecule ligand

Varin, Thibault, Godfrey, Alexander G., Masquelin, Thierry, Nicolaou, Christos A., Evans, David A., Vieth, Michal

Journal:

Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics

Année:

2015

Langue:

english

Fichier:

PDF, 807 KB

english, 2015

18

Solid-Phase Synthesis of Pyrimido[4,5- d ]pyrimidine-2,4(1 H ,3 H )-diones

Graveleau, Nadège, Masquelin, Thierry

Journal:

Année:

2003

Langue:

english

Fichier:

PDF, 68 KB

english, 2003

19

Coccidiostatic Agents: Synthesis of some Analogs of (±)-Frenolicin B

Masquelin, Thierry, Hengartner, Urs, Streith, Jacques

Journal:

Année:

1995

Fichier:

PDF, 674 KB

1995

20

A New Approach to the Synthesis of N-Protected 2- and 5-Substituted 3-Halopyrroles

Masquelin, Thierry, Obrecht, Daniel

Journal:

Année:

1995

Fichier:

PDF, 990 KB

1995

21

Identification of Phenoxyalkylbenzimidazoles with Antitubercular Activity

Chandrasekera, N. Susantha, Alling, Torey, Bailey, Mai A., Files, Megan, Early, Julie V., Ollinger, Juliane, Ovechkina, Yulia, Masquelin, Thierry, Desai, Prashant V., Cramer, Jeffrey W., Hipskind, Phi

Journal:

Journal of Medicinal Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 671 KB

english, 2015

22

Imidazo[1,2- a ]pyridine-3-carboxamides are Active Antimicrobial Agents of Mycobacterium avium Infection In Vivo

Moraski, Garrett C., Cheng, Yong, Cho, Sanghyun, Cramer, Jeffrey W., Godfrey, Alexander, Masquelin, Thierry, Franzblau, Scott G., Miller, Marvin J., Schorey, Jeffery

Journal:

Antimicrobial Agents and Chemotherapy

Année:

2016

Langue:

english

Fichier:

PDF, 758 KB

english, 2016

23

Novel Solution- and Solid-Phase Syntheses of Heterocyclic Systems

Cabon, Gaelle, Gaucher, Berangere, Gegout, Aline, Heulle, Sophie, Masquelin, Thierry

Journal:

CHIMIA International Journal for Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 134 KB

english, 2003

24

Prediction of drug penetration in tuberculosis lesions

Sarathy, Jansy Passiflora, Zuccotto, Fabio, Ho, Hsin-Pin, Sandberg, Lars, Via, Laura E, Marriner, Gwendolyn A., Masquelin, Thierry, Wyatt, Paul G., Ray, Peter Christopher, Dartois, Veronique

Journal:

ACS Infectious Diseases

Année:

2016

Langue:

english

Fichier:

PDF, 810 KB

english, 2016

25

The synthesis and evaluation of triazolopyrimidines as anti-tubercular agents

Zuniga, Edison S., Korkegian, Aaron, Mullen, Steven, Hembre, Erik J., Ornstein, Paul L., Cortez, Guillermo, Biswas, Kallolmay, Kumar, Naresh, Cramer, Jeffrey, Masquelin, Thierry, Hipskind, Philip A.,

Journal:

Bioorganic & Medicinal Chemistry

Année:

2017

Langue:

english

Fichier:

PDF, 1.05 MB

english, 2017

26

In Vitro Evaluation of Novel Nitazoxanide Derivatives against Mycobacterium tuberculosis

Odingo, Joshua, Bailey, Mai A., Files, Megan, Early, Julie V., Alling, Torey, Dennison, Devon, Bowman, Julie, Dalai, Suryakanta, Kumar, Naresh, Cramer, Jeffrey, Masquelin, Thierry, Hipskind, Philip A.

Journal:

Année:

2017

Langue:

english

Fichier:

PDF, 879 KB

english, 2017

27

Imidazopyridine compounds inhibit mycobacterial growth by depleting ATP levels

O'Malley, Theresa, Alling, Torey, Early, Julie V., Wescott, Heather A., Kumar, Anuradha, Moraski, Garrett C., Miller, Marvin J., Masquelin, Thierry, Hipskind, Philip A., Parish, Tanya

Journal:

Antimicrobial Agents and Chemotherapy

Année:

2018

Langue:

english

Fichier:

PDF, 933 KB

english, 2018

28

Synthesis and Evaluation of the 2-Aminothiazoles as Anti-Tubercular Agents

Kesicki, Edward A., Bailey, Mai A., Ovechkina, Yulia, Early, Julie V., Alling, Torey, Bowman, Julie, Zuniga, Edison S., Dalai, Suryakanta, Kumar, Naresh, Masquelin, Thierry, Hipskind, Philip A., Oding

Journal:

Année:

2016

Langue:

english

Fichier:

PDF, 930 KB

english, 2016

29

A High-Throughput Screen against Pantothenate Synthetase (PanC) Identifies 3-Biphenyl-4-Cyanopyrrole-2-Carboxylic Acids as a New Class of Inhibitor with Activity against Mycobacterium tuberculosis

Kumar, Anuradha, Casey, Allen, Odingo, Joshua, Kesicki, Edward A., Abrahams, Garth, Vieth, Michal, Masquelin, Thierry, Mizrahi, Valerie, Hipskind, Philip A., Sherman, David R., Parish, Tanya, Torrelle

Journal:

Année:

2013

Langue:

english

Fichier:

PDF, 1.22 MB

english, 2013

30

Identification of Morpholino Thiophenes as Novel Mycobacterium tuberculosis Inhibitors, Targeting QcrB

Cleghorn, Laura A. T., Ray, Peter, Odingo, Joshua, Kumar, Anuradha, Wescott, Heather, Korkegian, Aaron, Masquelin, Thierry, L. Moure, Abraham, Wilson, Caroline, Davis, Susan Helen, Huggett, Margaret J

Journal:

Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 942 KB

english, 2018

31

Identification of compounds with pH-dependent bactericidal activity against Mycobacterium tuberculosis

Early, Julie, Ollinger, Juliane, Darby, Crystal, Alling, Torey, Mullen, Steven, Casey, Allen, Gold, Ben, Ochoada, Jason, Wiernicki, Todd, Masquelin, Thierry, Nathan, Carl F., Hipskind, Philip, Parish,

Journal:

ACS Infectious Diseases

Année:

2018

Langue:

english

Fichier:

PDF, 1.08 MB

english, 2018